TargetVoltage-gated sodium channel Nav1.5 cardiac isoform(Canis lupus familiaris)
Gilead Sciences
Curated by ChEMBL
Gilead Sciences
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of canine ventricular myocytes Nav 1.5 assessed as reduction in ATX-2 induced late channel current by manual single-patch clamp assayMore data for this Ligand-Target Pair